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27 articles for University of Cagliari


The following articles (labelled with PubMed ID or TBD) are for your review
PMIDArticle TitlePublishedDeposition
32435395 New Dihydrothiazole Benzensulfonamides: Looking for Selectivity toward Carbonic Anhydrase Isoforms I, II, IX, and XII. 14-MAY-2020 12-AUG-2021
31422224 Synthesis and in vitro evaluation of piperazinyl-ureido sulfamates as steroid sulfatase inhibitors. 15-NOV-2019 25-FEB-2021
31472471 Structure-activity relationship with pyrazoline-based aromatic sulfamates as carbonic anhydrase isoforms I, II, IX and XII inhibitors: Synthesis and biological evaluation. 15-NOV-2019 21-FEB-2021
31442684 Chromenone derivatives as a versatile scaffold with dual mode of inhibition of HIV-1 reverse transcriptase-associated Ribonuclease H function and integrase activity. 15-NOV-2019 21-FEB-2021
30344915 Tuning the Dual Inhibition of Carbonic Anhydrase and Cyclooxygenase by Dihydrothiazole Benzensulfonamides. 11-OCT-2018 18-AUG-2020
30034608 Targeting Tumor Associated Carbonic Anhydrases IX and XII: Highly Isozyme Selective Coumarin and Psoralen Inhibitors. 12-JUL-2018 14-AUG-2020
28535469 Novel propanamides as fatty acid amide hydrolase inhibitors. 18-AUG-2017 02-JUL-2020
28835790 -Acylbenzenesulfonamide Dihydro-1,3,4-oxadiazole Hybrids: Seeking Selectivity toward Carbonic Anhydrase Isoforms. 10-AUG-2017 23-APR-2020
26995529 2-Phenylbenzofuran derivatives as butyrylcholinesterase inhibitors: Synthesis, biological activity and molecular modeling. 15-APR-2016 08-AUG-2017
26233435 Synthesis of sulfonamides incorporating piperazinyl-ureido moieties and their carbonic anhydrase I, II, IX and XII inhibitory activity. 17-AUG-2015 27-NOV-2016
26233796 Synthesis and carbonic anhydrase I, II, IX and XII inhibitory activity of sulfamates incorporating piperazinyl-ureido moieties. 31-AUG-2015 16-NOV-2016
26073006 New 4-[(3-cyclohexyl-4-aryl-2,3-dihydro-1,3-thiazol-2-ylidene)amino]benzene-1-sulfonamides, synthesis and inhibitory activity toward carbonic anhydrase I, II, IX, XII. 06-JUL-2015 11-NOV-2016
25728026 (3Z)-3-(2-[4-(aryl)-1,3-thiazol-2-yl]hydrazin-1-ylidene)-2,3-dihydro-1H-indol-2-one derivatives as dual inhibitors of HIV-1 reverse transcriptase. 13-MAR-2015 23-APR-2016
24589511 Synthesis and carbonic anhydrase I, II, IX and XII inhibition studies of 4-N,N-disubstituted sulfanilamides incorporating 4,4,4-trifluoro-3-oxo-but-1-enyl, phenacylthiourea and imidazol-2(3H)-one/thione moieties. 31-MAR-2014 07-FEB-2015
21216504 Opioid bifunctional ligands from morphine and the opioid pharmacophore Dmt-Tic. 25-JAN-2011 04-JAN-2013
16942034 Effect of lysine at C-terminus of the Dmt-Tic opioid pharmacophore. 31-AUG-2006 08-DEC-2012
12459023 Potent delta-opioid receptor agonists containing the Dmt-Tic pharmacophore. 02-DEC-2002 27-NOV-2012
22014547 Ungeremine effectively targets mammalian as well as bacterial type I and type II topoisomerases. 07-NOV-2011 21-JUL-2012
21777011 3-Acetyl-2,5-diaryl-2,3-dihydro-1,3,4-oxadiazoles: a new scaffold for the selective inhibition of monoamine oxidase B. 15-SEP-2011 23-MAR-2012
7664823 Modulation of [35S]TBPS binding by ligands with preferential affinity for benzodiazepine BZ1 sites in the cerebral cortex of newborn and adult rats. 23-XXX-1995 23-DEC-2011
20637637 Role of 2',6'-dimethyl-l-tyrosine (Dmt) in some opioid lead compounds. 09-AUG-2010 19-MAR-2011
20143779 Synthesis and evaluation of paracetamol esters as novel fatty acid amide hydrolase inhibitors. 04-MAR-2010 01-SEP-2010
19642675 Influence of the side chain next to C-terminal benzimidazole in opioid pseudopeptides containing the Dmt-Tic pharmacophore. 03-SEP-2009 27-AUG-2010
18680274 Further studies on lead compounds containing the opioid pharmacophore Dmt-Tic. 25-AUG-2008 11-JAN-2010
16107162 From the potent and selective mu opioid receptor agonist H-Dmt-d-Arg-Phe-Lys-NH(2) to the potent delta antagonist H-Dmt-Tic-Phe-Lys(Z)-OH. 18-AUG-2005 10-NOV-2009
17339114 Further studies on the effect of lysine at the C-terminus of the Dmt-Tic opioid pharmacophore. 02-APR-2007 10-NOV-2009
16366592 Conversion of the potent delta-opioid agonist H-Dmt-Tic-NH-CH(2)-bid into delta-opioid antagonists by N(1)-benzimidazole alkylation(1). 21-DEC-2005 10-NOV-2009